Supply 99.9% Purity Tianeptine Sulfate CAS:1224690-84-9

Quick Details

• CasNo： 1224690-84-9
• Molecular Formula： C42H56Cl2N4O14S3
• Appearance： White Powder
• Delivery Time： 3days after we receive the payment
• Throughput： 1000|Kilogram|Month
• Purity： 99.5%

High Quality Tianeptine Sulfate powder

Tianeptine has been in use for a few decades as an effective treatment for depression. Still, a certain controversial fact has emerged in 2014. It’s triggered its ban in several in several countries including the UK.

A 2014 study found that tianeptine is a mu-opioid receptor full agonist. This explains its opioid-like effects which mostly occur when taking extremely high doses.

Still, even though it acts on the same receptors, tianeptine combines well with morphine. This is to prevent respiratory depression associated with opioids. 

Some of its antidepressant effects occur due to the alteration of glutamate receptor activity, namely the AMPA and NMDA receptors, as well as through the release of BDNF (brain-derived neurotrophic factor) which affects neuroplasticity.

Furthermore, tianeptine enhances the mesolimbic release of dopamine by potentiating the D2 and D3 receptors. 

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Tianeptine sodium vs. Tianeptine sulfate

When thinking of tianeptine sulfate vs sodium, choosing the right one for you depends on several factors. Some prefer one over the other according to onset, duration, bioavailability, taste and degradation rate.

Onset/Duration – Tianeptine sulfate takes a few hours to kick in. Still, it’ll last a whole day, thus only necessitating a single daily dose. Tianeptine sodium kicks in faster and is three to four times more potent. Also, you should take tianeptine sodium four times a day for its effects to be continuously felt.

Bioavailability – Tianeptine sulfate has a higher solubility in water, thus increasing its bioavailability.

Stability – Tianeptine sodium rapidly degrades after you open the seal due to moisture and exposure to light.

Taste – Tianeptine sulfate is almost insipid, while tianeptine sulfate has a bitter taste.

From a medical point of view, tianeptine sulfate is better for somebody undergoing treatment. That’s because the risk of ineffective treatment caused by skipping doses significantly decreases when the user only needs one daily dose.

Also, tianeptine sodium provides an immediately noticeable increase in energy and motivation. Tianeptine sulfate is not as energizing. That’s because of one would need a higher dose and its onset is a lot slower.

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